专利详细信息
专利号 | EP2481726A3 |
专利标题 | Crystal forms of saxagliptin and processes for preparing same |
专利权人 | BRISTOL-MYERS SQUIBB COMPANY; |
发明人 | Gougoutas, Jack Z;Malley, Mary F;Dimarco, John D;Yin, Xiaotian S;Wei, Chenkou;Yu, Jurong;Vu, Truc Chi;Jones, Gregory Scott;Savage, Scott A; |
申请号 | EP20120164711 |
申请日 | 2008/4/18 |
公开日 | 2014/3/5 |
优先权号 | |
IPC | C07D20952000; |
专利类型 | |
法律状态查询 | 查看法律状态 |
Physical crystal structures of a compound of the formula (I): are provided including the free base monohydrate thereof (form H-1) and the hydrochloric acid salt thereof including hydrochloric acid salt containing 0.75 equivalent of H2O (form H0.75-3) and hydrochloric acid salt containing 2 equivalents of H2O (form H2-1) and hydrochloric acid salt Pattern P-5 preferably in substantially pure form and other forms as described herein pharmaceutical compositions containing structures of compound I or IA processes for preparing same intermediates used in preparing same and methods of treating diseases such as diabetes using such structures.
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